発表論文
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主な発表論文
2012年
- Nagaoka K, Hanioka N, Ikushiro S, Yamano S, Narimatsu S.
The effects of N-glycosylation on the glucuronidation of zidovudine and morphine by UGT2B7 expressed in HEK293 cells.
Drug Metab Pharmacokinet., 27, 388-397 (2012)
- Uchihashi S, Nishikawa M., Sakaki T., Ikushiro S.
The critical role of amino acid residue at position 117 of mouse UDP-glucuronosyltransfererase 1a6a and 1a6b in resveratrol glucuronidation.
J.Biochem. 152, 331-340 (2012)
- Zhang H., Patana A., Mackenzie PI., Ikushiro S., Goldman A., Finel M.
Human UDP-glucuronosyltransferase expression in insect cells: ratio of active to inactive recombinant proteins and the effects of a C-terminal his-tag on glucuronidation kinetics.
Drug Metabolism and Disposition, 40, 1935-1944 (2012)
- Yasuda K, Ikushiro S, Wakayama S, Itoh T, Yamamoto K.,Kamakura M, Munetsuna E, Ohta M, Sakaki T.
Comparison of metabolism of sesamin and episesamin by drug-metabolizing enzymes in human liver.
Drug Metabolism and Disposition, 40, 1917-1926 (2012)
- Kato Y., Tamaki S., Haraguchi K.,Ikushiro S., Sekimoto M., Ohta C., Endo T., Koga N., Yamada S., Degawa M.
Comparative study on 2,2',4,5,5'-pentachlorobiphenyl-mediated decrease in serum thyroxine level between C57BL/6 and its transthyretin-deficient mice.
Toxicology and Applied Pharmacology, 263, 323-329 (2012)
- Yasuda K, Ikushiro S, Kamakura M, Takano M, Saito N, Kittaka A, Chen TC, Ohta M, Sakaki T.
Human cytochrome P450-dependent differential metabolism among three 2α-substituted-1α,25-dihydroxyvitamin D3 analogs.
J Steroid Biochem Mol Biol., 133, 84-92 (2012)
- Sawada D, Tsukuda Y, Yasuda K, Sakaki T, Saito H, Takagi K, Takenouchi K, Chen TC, Reddy GS, Kittaka A.
Synthesis and biological activities of 1α,4α,25- and 1α,4β,25-trihydroxyvitamin D3 and their metabolism by human CYP24A1 and UDP-glucuronosyltransferase.
Chem Pharm Bull (Tokyo), 60, 1343-1346 (2012)
- Kawamura-Konishi Y, Watanabe N, Saito M, Nakajima N, Sakaki T, Katayama T, Enomoto T.
Isolation of a new phlorotannin, a potent inhibitor of carbohydrate-hydrolyzing enzymes, from the brown alga Sargassum patens.
J Agric Food Chem. 6, 5565-5570 (2012)
- Kittaka A, Yoshida A, Chiang KC, Takano M, Sawada D, Sakaki T, Chen TC.
Potent 19-norvitamin D analogs for prostate and liver cancer therapy.
Future Med Chem. 4, 2049-2065 (2012)
- Yasuda K, Sakaki T.
How is sesamin metabolised in the human liver to show its biological effects?
Expert Opin Drug Metab Toxicol. 8, 93-102, Review (2012)
- Chen TC, Sakaki T, Yamamoto K, Kittaka A.
The roles of cytochrome P450 enzymes in prostate cancer development and treatment.
Anticancer Res. 32, 291-298, Review (2012)
- Sakaki T.
Practical application of cytochrome P450.
Biol Pharm Bull., 35, 844-849, Review (2012)
- 鎌倉昌樹
ミツバチの女王蜂分化を誘導する因子ロイヤラクチンの発見
生物の科学遺伝, 66, 82-88総説(2012)
- 鎌倉昌樹
ミツバチの女王蜂分化を誘導する因子ロイヤラクチンの発見
バイオサイエンスとインダストリー, 70, 115-119 総説(2012)
- 鎌倉昌樹
ミツバチの女王蜂分化を誘導する因子ロイヤラクチンの発見
生化学, 84, 994-1003 総説(2012)
- 鎌倉昌樹
ロイヤラクチンの発見からミツバチの生態解明へ
細胞工学, 31, 1166-1169 総説(2012)
- 鎌倉昌樹
ミツバチの女王蜂分化を誘導する因子ロイヤラクチンの発見
化学と生物, 50, 476-478 総説(2012)
- 鎌倉昌樹
ミツバチの幼虫を女王バチに成長させるタンパク質の発見
農林水産技術研究ジャーナル, 35, 53-56 総説(2012)
- 鎌倉昌樹
女王を育むロイヤラクチン
生命誌ジャーナル, 74,(オンライン版)、JT生命誌研究館 (2012)
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