発表論文

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主な発表論文

2015年

  1. Yasuda K, Ueno S, Ueda E, Nishikawa M, Takeda K, Kamakura M, Ikushiro S, Sakaki T.
    Influence of sesamin on CYP2C-mediated diclofenac metabolism: in vitro and in vivo analysis.
    Pharmacol Res Perspect. 3, e00174 (2015)
  2. Shirotani N, Togawa M, Ikushiro S, Sakaki T, Harada T, Miyagawa H, Matsui M, Nagahori H, Mikata K, Nishioka K, Hirai N, Akamatsu M.
    Identification and in silico prediction of metabolites of the model compound, tebufenozide by human CYP3A4 and CYP2C19.
    Bioorg Med Chem. 23, 6594-6601 (2015)
  3. Mano H, Nishikawa M, Yasuda K, Ikushiro S, Saito N, Takano M, Kittaka A, Sakaki T.
    Development of Novel Bioluminescent Sensor to Detect and Discriminate between Vitamin D Receptor Agonists and Antagonists in Living Cells.
    Bioconjug Chem., 26, 2038-2045 (2015)
  4. Bolla NR, Corcoran A, Yasuda K, Chody?ski M, Krajewski K, Cmoch P, Marcinkowska E, Brown G, Sakaki T, Kutner A.
    Synthesis and evaluation of geometric analogs of 1α,25-dihydroxyvitamin D2 as potential therapeutics.
    J Steroid Biochem Mol Biol. pii: S0960-0760(15)30057-1 (2015)
  5. Takano M, Yasuda K, Higuchi E, Tohyama E, Takeuchi A, Sakaki T, Kittaka A.
    Synthesis, metabolism, and biological activity of 2-[3-(tetrazolyl)propyl]-1α,25-dihydroxy-19-norvitamin D3.
    J Steroid Biochem Mol Biol. pii: S0960-0760(15)30029-7 (2015)
  6. Yasuda K, Iwanaga Y, Ogawa K, Mano H, Ueno S, Kimoto S, Ohta M, Kamakura M, Ikushiro S, Sakaki T.
    Human hepatic metabolism of the anti-osteoporosis drug eldecalcitol involves sterol C4-methyl oxidase.
    Pharmacol Res Perspect., 3, e00120 (2015)
  7. Watanabe KP, Kawai YK, Nakayama SM, Ikenaka Y, Mizukawa H, Takaesu N, Ito M, Ikushiro SI, Sakaki T, Ishizuka M.
    Partial cloning of CYP2C23a genes and hepatic protein expression in eight representative avian species.
    Journal of Veterinary Pharmacology and Therapeutics, 38, 190-195 (2015)
  8. Takano M, Sawada D, Yasuda K, Nishikawa M, Takeuchi A, Takagi K, Horie K, Reddy GS, Chen TC, Sakaki T, Kittaka A.
    Synthesis and metabolic studies of 1α,2α,25-, 1α,4α,25- and 1α,4β,25-trihydroxyvitamin D3.
    J Steroid Biochem Mol Biol. 148, 34-37 (2015)
  9. Maruo Y, Behnam M, Ikushiro S, Nakahara S, Nouri N, Salehi M.
    Two Different UGT1A1 Mutations causing Crigler-Najjar Syndrome types I and II in an Iranian Family.
    J Gastrointestin Liver Dis. 24, 523-526 (2015)
  10. 榊利之
    代謝研究に基づくビタミンD作用メカニズムの再考
    生化学, 87, 438-444 (2015)
  11. 安田佳織、岩永由麻、小川和亮、真野寛生、上野千来、木本周太朗、太田美穂、鎌倉昌樹、生城真一、榊利之
    骨粗鬆症治療薬エルデカルシトールの代謝にメチルステロール酸化酵素SC4MOLが関与する
    ビタミン, 89, 492-494 (2015)

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